Khoom Description
Olaparib yog dab tsi?
Olaparib hmoovyog chemical raw khoom. Nws lub npe tshuaj yog 4-[(3-{[4-}(6-Fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]methyl}phenyl)carbamoyl]-2-methylbenzoic acid, chemical formula 3 F4N4H2 yog C24H2. Tsis muaj. yog763113-22-0. Nws belongs rau PARP (poly (ADP-ribose) polymerase) inhibitor chav kawm, uas tuaj yeem cuam tshuam kev ua haujlwm ntawm PARP enzymes hauv hlwb. PARP enzymes yog cov enzymes tseem ceeb rau kev kho DNA puas. Nws cov qauv tshuaj muaj ntau pawg ua haujlwm xws li benzene rings, oxygen heterocycles, thiab pyridine rings, nrog cov fluorine atom ntawm cov pa heterocycle. Cov yam ntxwv ntawm cov tshuaj no ua rau nws xaiv tau zoo thiab muaj kev sib raug zoo rau cov hom phiaj PARP enzymes.
Olaparib APIyog qhov ncauj PARP (polymerase RNA polymerase) inhibitor siv los kho qee yam kab mob BRCA gene mutation-associated disease. Hauv qab no yog nws cov keeb kwm kev loj hlob thiab kev cia siab:
Kev Tshawb Nrhiav thiab kev loj hlob: Olaparib, Ameslikas tsim los ntawm AstraZeneca, tau pom zoo los ntawm US FDA hauv 2014, dhau los ua thawj cov tshuaj tau txais kev pom zoo ua lag luam rau PARP inhibitor. Nws txoj kev txhim kho tau dhau los ntawm ntau theem los ntawm kev tshuaj xyuas tshuaj mus rau kev sim tshuaj.
Kev siv tam sim no: Olaparib tau dhau los ua ib qho ntawm cov tshuaj tseem ceeb siv los kho qee yam kab mob BRCA hloov pauv. Tib lub sijhawm, qee cov kws tshawb fawb tab tom kawm txog nws cov ntawv thov hauv kev kho mob rau lwm yam kab mob.
Kev Pom Zoo: Nrog rau kev kawm ntxiv txog cov txheej txheem ntawm kev ua ntawm PARP inhibitors, daim ntawv thov ntawm Olaparib thiab cov tshuaj zoo sib xws tseem muaj kev cia siab, tshwj xeeb tshaj yog nyob rau hauv kev kho mob ntawm qee yam kab mob ntsig txog BRCA noob txawv txav. Nyob rau tib lub sijhawm, kev txhim kho ntawm nws cov kev mob tshwm sim thiab kev ua siab ntev kuj yuav yog ib qho ntawm cov lus qhia tseem ceeb ntawm kev txhim kho yav tom ntej, txhawm rau txhim kho tus nqi ciaj sia thiab kev kho mob ntawm cov neeg mob.
Cov ntaub ntawv tseem ceeb:
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Khoom npe |
Olaparib |
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tshuaj npe |
4-[(3-{[{2}}(6-Fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]methyl}phenyl)carbamoyl]-2-methylbenzoic acid |
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CAS |
763113-22-0 |
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MF |
C24H23FN4O3 |
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MW |
434.46 |
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EINECS |
642-941-5 |
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MDL Nr. |
TIAB SA 13185161 |
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Purity |
99 feem pua |
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Kev ruaj ntseg |
Nyob ruaj khov nyob rau hauv kev pom zoo cia. |
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solubility |
ruaj khov |
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Daim ntawv thov |
Qib tshuaj los yog siv rau kev tshawb fawb. |
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Ntim |
Raws li koj qhov kev thov |
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Cia |
Chav ntsuas kub. |
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Cov qauv qauv |
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Cov qauv zoo:
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KEV KAWM |
STANDARD |
TSEEM CEEB |
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Qhov tshwm sim |
hmoov dawb |
hmoov dawb |
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Kev txheeb xyuas |
IR |
Ua raws |
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HPLC |
Ua raws |
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Dej |
Tsawg dua lossis sib npaug rau 0.5 feem pua |
0.35 feem pua |
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Residue ntawm ignition |
Tsawg dua lossis sib npaug rau 0.1 feem pua |
0.07 feem pua |
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Residual Solvents |
Ethanol Tsawg dua lossis sib npaug rau 0.5 feem pua |
0.080 feem pua |
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Dichloromethane Tsawg dua lossis sib npaug rau 0.06 feem pua |
0.030 feem pua |
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Hais txog impurity |
Ib qho impurity Tsawg dua lossis sib npaug rau 0.1 feem pua |
0.07 feem pua |
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Tag nrho impurity Tsawg dua lossis sib npaug rau 0.5 feem pua |
0.11 feem pua |
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HPLC kev xeem |
98. 0-102 {2}} feem pua |
99.4% ua |
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Xaus |
Ua raws li Enterprise Standard |
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Tsuas yog siv rau kev lag luam lossis kev tshawb fawb, tsis yog khoom siv rau ib tus neeg twg!
khaws cia
Cov xwm txheej cia rauOlaparib hmoovyog ib qho tseem ceeb heev rau nws zoo thiab stability. Nov yog cov xwm txheej khaws cia:
Kub: Nws yuav tsum tau khaws cia nyob rau hauv thaj tsam ntawm 2-8 degrees Celsius. Tsis txhob khaws cia rau hauv qhov chaw kub kub.
Humidity: Nws kuj tseem ceeb rau cov av noo. Nws yuav tsum tau muab cia rau hauv qhov chaw qhuav, thiab nyob rau hauv ib lub thawv kaw kom tsis txhob ya raws.
Ntim thiab sealing: Khaws cia rau hauv nws qhov ntim thawj thiab xyuas kom meej tias lub hnab ntim khoom lossis lub raj mis tsis zoo thiab kaw zoo. Qhov no yuav pab tiv thaiv kom tsis txhob ya raws thiab huab cua nkag.
pls nco ntsoov cov kev cia tshwj xeeb yuav txawv nyob ntawm tus qauv thiab cov chaw tsim khoom. Ua ntej khaws cia thiab siv Olaparib hmoov, nws raug nquahu kom sab laj nrog cov chaw tsim khoom cov lus qhia tshwj xeeb lossis nrhiav tswv yim los ntawm kws kho mob lossis kws muag tshuaj.
Packing & shipping
Ntim:
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1 ~ 2 kg |
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2-10kg |
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10-25kg |
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Shipping:
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Tsawg dua los yog sib npaug li 50 kg |
Los ntawm kev nthuav qhia qhov rooj rau qhov rooj Fedex, DHL, UPS, TNT, EMS thiab lwm yam. Ceev thiab yooj yim |
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50kg-200kg |
Los ntawm huab cua Ceev thiab pheej yig |
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Ntau tshaj lossis sib npaug li 200kg |
Los ntawm hiav txwv Txoj kev pheej yig tshaj |
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Los yog raws li koj yuav tsum tau xaiv txoj kev pheej yig tshaj los yog ceev. |
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Lub sijhawm them nyiaj

Vim li cas thiaj xaiv Xi'an Yihui?
Raws li Olaparib tsum, Xi'an Yihui muaj cov hauv qab no zoo:
Kev tsim khoom nplua nuj thiab kev paub txog kev paub: peb yog cov kws tshaj lij kev lag luam koom nrog kev tshawb fawb, kev tsim khoom, thiab kev muag khoom ntawm cov tshuaj intermediates thiab cov ntaub ntawv raw. peb muaj kev paub nplua nuj thiab kev paub txog kev tsim khoom ntawm Olaparib.
High-quality: peb ua raws li lub hauv paus ntsiab lus ntawm kev ua tau zoo ua ntej, thiab cov khoom tsim tau ruaj khov nyob rau hauv zoo, siab purity, thiab zoo. peb tau dhau ntau daim ntawv pov thawj zoo.
Lub peev xwm tsim tau yooj yim thiab lub voj voog xa khoom sai: peb muaj peev xwm tsim tau yooj yim thiab tuaj yeem kho cov phiaj xwm tsim khoom raws li cov neeg siv khoom xav tau, ua kom lub voj voog luv luv, thiab ua tau raws li cov neeg siv khoom xav tau.
Kev pabcuam zoo rau cov neeg siv khoom: peb muab qhov tseem ceeb rau cov neeg siv khoom xav tau thiab kev tawm tswv yim, thiab muaj pab pawg neeg ua haujlwm tshaj lij uas muab kev pabcuam zoo, raws sijhawm, thiab cov kev pabcuam zoo ua ntej muag thiab kev pabcuam tomqab muag los muab cov neeg siv khoom zoo dua thiab kev pabcuam.

Xi 'an Yihui tuam txhab muag khoom, khoom siv ntau lawm

Xi'an Yihui tuam txhab muaj qib siab ntawm kev tshawb fawb thiab kev txhim kho muaj peev xwm

Xi 'an Yihui Company's Advanced ntau lawm cov cuab yeej thiab tshuab

Zoo meej kev pab cuam tom qab muag
Hauv kev xaus, raws li tus neeg muag khoom ntawmOlaparib hmoov, Xi'an Yihui muaj kev paub ntau lawm thiab kev paub, cov khoom zoo, muaj peev xwm ua tau zoo, thiab cov neeg siv khoom zoo, uas tuaj yeem muab kev txhawb nqa zoo dua thiab kev pabcuam rau cov neeg siv khoom.
Cim npe nrov: Tuam Tshoj olaparib hmoov manufacturers, lwm tus neeg, Hoobkas


















