Khoom Description
Varenicline tartrate yog dab tsi?
Varenicline tartrate hmoov, kuj hu ua tartrate ntsev. Nws lub npe tshuaj yog (1,2,3,4-tetrahydro-2-methyl-3-(3-pyridyl)-1,5-benzodiazepin{{ 9}}yl) (1,4-dihydroxy-2,3,5,6-tetraoxy-hexane-1,1,4,4-tetrayl) dipyrophosphate . Nws yog dawb mus rau dawb crystalline hmoov, nws yog soluble hauv dej thiab methanol ntawm chav tsev kub. Nws cov mis molecular yog C13H13N3.C4H6O6P2, nws cov txheeb ze molecular hnyav yog 361.3 g / mol, CAS tus lej yog375815-87-5. Nws cov tshuaj pharmacological ntawm kev ua haujlwm suav nrog kev khi rau 4 2 nicotinic acetylcholine receptors ntawm cov neurons, ua kom cov receptors no, thiab nce dopamine tso tawm, ua rau cov teebmeem zoo li nicotine. nws tuaj yeem txo qhov kev haus luam yeeb nyob hauv cov neeg haus luam yeeb los ntawm kev ua raws li cov txiaj ntsig ntawm nicotine thaum txo cov tsos mob tshem tawm cuam tshuam nrog kev txiav luam yeeb. nws txoj kev loj hlob tau pib thaum xyoo 1990s thaum Pfizer nqis peev ntau los nrhiav kev haus luam yeeb zoo dua. Lawv cov kev tshawb fawb tau tsom mus rau nicotinic receptors, vam tias yuav tsim cov tshuaj uas tuaj yeem ua raws li nicotine cov teebmeem thiab txo cov tsos mob tshem tawm. Tom qab kev sim ntau thiab kev sim, cov kws tshawb fawb tau ua tiav tiavVarenicline tartrate API. Cov tshuaj tau pom zoo los ntawm US FDA xyoo 2006 thiab tom qab ntawd tau pom zoo siv rau ntau lub tebchaws. Txij li thaum nws tau pom zoo, nws tau pom tias yog ib qho tshuaj tiv thaiv kev haus luam yeeb tau zoo, txo qis kev haus luam yeeb thiab txo qis cov tsos mob. Txawm hais tias qee qhov kev tsis sib haum xeeb thiab cov lus ceeb toom ntawm cov xwm txheej tsis zoo, nws tseem yog qhov kev xaiv zoo tshaj plaws rau ntau tus neeg uas xav txiav luam yeeb. Zuag qhia tag nrho, txoj kev loj hlob ntawm Varenicline tartrate koom nrog xyoo ntawm kev tshawb fawb thiab kev loj hlob, thaum kawg ua tau zoo heev thiab dhau los ua ib qho kev kho tseem ceeb rau kev haus luam yeeb.
Cov ntaub ntawv tseem ceeb:
|
Khoom npe |
Varenicline tartrate |
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Lwm lub npe |
CS-291;Champix;Pidifix330;Pidifix-330;CP 526555-18;Unii-82269asb48;Champix tartrate;Chantix tartrate;Varniclan tartrate |
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CAS |
375815-87-5 |
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MF |
C17H19N3O6 |
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MW |
361.35 |
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EINECS |
638-780-5 |
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MDL Nr. |
TIAB SA 08460603 |
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Purity |
99% |
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Kev ruaj ntseg |
ruaj khov thaum khaws cia rau hauv cov xwm txheej tsim nyog. |
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solubility |
Me ntsis soluble hauv dej |
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Daim ntawv thov |
Qib tshuaj los yog siv rau kev tshawb fawb. |
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Ntim |
Raws li koj qhov kev thov |
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Cia |
Chav ntsuas kub. |
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Cov qauv qauv |
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Cov qauv zoo:
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Yam khoom |
Txuj |
Cov txiaj ntsig |
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Qhov tshwm sim |
Dawb kom tawm daj hmoov |
Ua raws |
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Purity |
Ntau dua lossis sib npaug li 96% |
99.06% |
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Tag nrho impurities |
1.0% Max. |
0.45% |
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Singl impurities |
0.5.% Max. |
0.33% |
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Poob rau ziab |
0.5% Max. |
0.30% |
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Tshauv |
0.5% Max. |
0.31% |
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Kev txheeb xyuas |
NMR |
Ua raws |
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Xaus |
Mus txog Tus Qauv |
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Tsuas yog siv rau kev lag luam lossis kev tshawb fawb, tsis yog khoom siv rau ib tus neeg twg!
Kev ruaj ntseg & Cia
Varenicline tartrate hmoovNws kuj yog qhov ruaj khov, tab sis nyob rau hauv qee qhov xwm txheej, nws yuav raug degradation lossis decomposition. Nws stability tuaj yeem piav raws li hauv qab no:
Thermal stability: nws yog qhov ruaj khov ntawm chav tsev kub, tab sis nws tuaj yeem ua rau ib nrab degradation nyob rau hauv qhov kub thiab txias. Ntawm 60 degree, nws muaj kev ruaj ntseg zoo, thiab tom qab muab cia rau hauv chav tsev kub rau 24 lub hlis, nws qhov zoo tshaj 98%.
Lub teeb ruaj khov: nws yog qhov ruaj khov rau lub teeb, tab sis nws maj mam poob kev ua haujlwm thaum raug lub teeb muaj zog thiab hluav taws xob ultraviolet. Yog li ntawd, nws yuav tsum tau tiv thaiv los ntawm raug rau lub teeb muaj zog thiab ultraviolet hluav taws xob thaum lub sij hawm tsim thiab cia.
Oxidative stability: nws muaj qhov zoo oxidation stability, nws yuav degraded yog tias raug oxidants pom tseeb (xws li hydrogen peroxide thiab Potassium permanganate).
Acid-alkali stability: nws yog rhiab rau acid-alkali ib puag ncig, thiab khaws cia rau hauv ib puag ncig acidic lossis alkaline yuav ua rau degradation.
Hauv cov ntsiab lus, txhawm rau ua kom zoo thiab ruaj khov, nws yuav tsum raug tiv thaiv los ntawm qhov kub thiab txias, lub teeb, oxidants, thiab acidic lossis alkaline ib puag ncig. Yuav tsum tau siv qhov chaw cia kom zoo, xws li dryness, tsis tshua muaj teeb, thiab tsis kub, yuav tsum tau siv. Thaum siv cov tshuaj, kuj yuav tsum tau them nyiaj mloog mus rau nws qhov zoo thiab hnub tas sij hawm kom tsis txhob cuam tshuam nws cov txiaj ntsig.
Cov cai cia khoom:
Cia qhov kub thiab txias: nws yuav tsum muab cia rau hauv qhov chaw qhuav, txias, thiab qhov cua zoo, nrog rau qhov ntsuas kub zoo tshaj yog 2 degree -8 degree . Khaws nws ntawm qhov ntsuas kub no tuaj yeem tswj tau qhov zoo thiab ruaj khov ntawm cov tshuaj thiab txuas ntxiv nws lub txee lub neej.
Kev tiv thaiv lub teeb: nws yog rhiab heev rau lub teeb, yog li cov thawv opaque yuav tsum tau siv los tiv thaiv cov tshuaj thaum lub sij hawm cia kom tsis txhob raug tshav ntuj ncaj qha los yog lub teeb muaj zog. Tsis txhob raug UV teeb.
Moisture-pov thawj: nws yog hygroscopic, yog li yuav tsum tsis txhob ya raws thaum khaws cia. Cov ntim ntim ntim thiab bioreagent desiccants tuaj yeem siv los tiv thaiv kom tsis txhob ya raws.
Tsis txhob khov: nws tsis tiv thaiv kom khov thiab tsis tuaj yeem khaws lossis thauj mus rau hauv qhov chaw khov, txwv tsis pub nws yuav ua rau cov tshuaj degradation thiab poob ntawm kev ua tau zoo.
Tsis txhob muaj kev vibration: nws yog hmoov, thiab yog tias nws dhau kev co lossis poob siab thaum khaws cia lossis kev thauj mus los, nws yuav tawg lossis deform, cuam tshuam rau nws qhov zoo thiab kev ua haujlwm.
Hauv cov ntsiab lus, txhawm rau tiv thaiv qhov zoo thiab ruaj khov, nws yuav tsum tau ua raws li kev khaws cia thiab kev thauj mus los. Tshwj xeeb, yam xws li qhov kub thiab txias, lub teeb, av noo, thiab kev vibration, ib zaug dhau qhov kev kam rau siab ntawm cov tshuaj, yuav ua rau cov tshuaj tsis ua haujlwm lossis degradation.
Packing & shipping
Ntim:
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1 ~ 2 kg |
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2-10kg |
|
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10-25kg |
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Shipping:
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Tsawg dua los yog sib npaug li 50 kg |
Los ntawm kev nthuav qhia qhov rooj rau qhov rooj Fedex, DHL, UPS, TNT, EMS thiab lwm yam. Ceev thiab yooj yim |
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50kg-200kg |
Los ntawm huab cua Ceev thiab pheej yig |
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Ntau tshaj lossis sib npaug li 200kg |
Los ntawm hiav txwv Txoj kev pheej yig tshaj |
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Los yog raws li koj yuav tsum tau xaiv txoj kev pheej yig tshaj los yog ceev.
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Lub sijhawm them nyiaj

Vim li cas thiaj xaiv Xi'an Yihui?
Hauv kev xaus, raws li tus kws tshaj lijVarenicline tartrate hmoovchaw tsim tshuaj paus, peb muaj advanced technology, scale kom zoo dua, qhov zoo tshaj plaws zoo, nplua nuj ntau lawm kev, thiab cov kev pab zoo heev. Cov txiaj ntsig zoo no yuav ua rau pebVarenicline tartrate APIsawv tawm hauv kev sib tw ua lag luam thiab yeej ntau tus neeg siv khoom ntseeg siab thiab kev txhawb nqa.

Xi 'an Yihui tuam txhab muag khoom, khoom siv ntau lawm

Xi'an Yihui tuam txhab muaj qib siab ntawm kev tshawb fawb thiab kev txhim kho muaj peev xwm

Xi 'an Yihui Company's Advanced ntau lawm cov cuab yeej thiab tshuab

Zoo meej kev pab cuam tom qab muag
Cim npe nrov: Tuam Tshoj varenicline tartrate hmoov manufacturers, lwm tus neeg, Hoobkas


















