Everolimus hmoov

Everolimus hmoov

Khoom npe: Everolimus
CAS: 159351-69-6
MF: C53H83NO14
MW: 958.22
Pob: 1g / hnab; 10g / hnab; 100g / hnab
Keeb kwm: Suav teb
Muaj peev xwm muab khoom: 50kg ib hlis
Qauv Muaj: Yog
Kev Them Nyiaj: T / T, LC lossis DA
Daim ntawv pov thawj: ISO9001, ISO22000, HACCP, HALAL, KOSHER
Muag tsis tau rau tib neeg

Tsham tam sim no
Khoom Taw qhia
Khoom Description

Everolimus yog dab tsi?

Everolimus hmoovyog ib qho tshuaj tiv thaiv kab mob hauv qhov ncauj uas ua rau lub hom phiaj taw qhia txoj hauv kev. Nws yog dawb los yog dawb crystalline hmoov nrog zoo thermal stability. Nws cov qauv tshuaj yog C53H83NO14, molecular hnyav yog 958.23 g / mol, thiab CAS tus lej yog159351-69-6. Solubility ntawm everolimus nce nrog nce pH. Nws feem ntau yog ua los ntawm cov tshuaj synthesis. Ua ntej, lub precursor compound C51H79NO13 yog synthesized, thiab ces deprotection thiab cyclization kauj ruam yog ua kom tau cov khoom everolimus. Nws yuav tsum tau muab cia rau hauv qhov chaw txias, qhuav, thiab tsis muaj teeb meem. Thaum lub sij hawm cia, nws yuav tsum tau tiv thaiv los ntawm noo noo, kub kub, thiab kev co.

Keeb kwm Discovery: nws yog Ameslikas tsim los ntawm Novartis, lub tuam txhab tshuaj Swiss. Cov kws tshawb fawb los ntawm lub tuam txhab pom nws los ntawm actinomycete Streptomyces hygroscopicus. Xyoo 1999, nws tau pom zoo rau kev lag luam los ntawm European Medicines Agency. Hauv xyoo 2009, nws tau pom zoo rau kev lag luam los ntawm FDA.

Daim ntawv thov tam sim no: nws tau dhau los ua ib qho ntawm cov tshuaj nquag siv hauv kev kho mob thiab muaj txiaj ntsig zoo hauv kev kho mob ntawm ntau yam kab mob.

Cov kev xav yav tom ntej: Nrog rau kev tshawb fawb ntxiv, cov kws tshawb fawb tau tshawb pom tias nws kuj muaj lwm yam tshuaj muaj txiaj ntsig, xws li tshuaj tua kab mob, tshuaj tiv thaiv kab mob, thiab tshuaj tiv thaiv kab mob fibrotic.Yog li ntawd, nws muaj kev thov dav dav hauv lwm qhov chaw. Nyob rau hauv lub neej yav tom ntej, nrog rau kev tshawb nrhiav ntxiv ntawm nws cov txheej txheem ntawm kev ua, nws yuav raug tshawb pom thiab siv rau kev kho mob ntau dua. Nyob rau tib lub sijhawm, nws kev sib xyaw nrog lwm cov tshuaj kuj tseem yog qhov kev tshawb fawb hotspot, uas yuav muab ntau txoj hauv kev rau kev nthuav dav nws daim ntawv thov ntau yam.

 

Cov ntaub ntawv tseem ceeb:

Khoom npe

Everolimus

tshuaj npe

(1R,9S,12S,15R,16E,18R,19R,21R,23S,24E,26E,28E,30S,32S,35R)-1,18-Dihydroxy-12-[(1R){1}S,35R, ethoxy) -3-methoxycyclohexyl]-1-methylethyl]-19,30-dimethoxy-15,17,21,23,29,35-}hexamethyl{35}},36-dioxa{{37}.conotahetricy. 44}},24,26,28-tetraene-2,3,10,14,{52}}pentone

CAS

159351-69-6

MF

C53H83NO14

MW

958.22

EINECS

621-003-9

MDL Nr.

TIAB SA 00929329

Purity

99 feem pua

Kev ruaj ntseg

ib tug kuj ruaj khov compound nrog zoo lub cev thiab tshuaj stability nyob rau hauv ib txwm cia tej yam kev mob. Nws feem ntau yog khaws cia rau hauv chav tsev kub hauv qhov chaw qhuav thiab zoo-ventilated, tiv thaiv los ntawm lub teeb thiab noo noo.

solubility

kuj tsis zoo soluble compound nyob rau hauv dej. Nws yog lipophilic heev, txhais tau hais tias nws muaj kev sib raug zoo rau lipid-raws li cov khoom siv xws li roj lossis roj, tab sis tsis tshua muaj solubility hauv aqueous media. Kev solubility ntawm Everolimus tuaj yeem cuam tshuam los ntawm cov khoom xws li pH, qhov kub thiab txias, thiab muaj lwm yam khoom ntxiv.

Daim ntawv thov

Qib tshuaj los yog siv rau kev tshawb fawb.

Ntim

Raws li koj qhov kev thov

Cia

Chav ntsuas kub.

Cov qauv qauv

159351-69-6

 

Cov qauv zoo:

 

Cov khoom

Specifications

Cov txiaj ntsig

Qhov tshwm sim

Dawb los yog dawb hmoov hmoov

Dawb hmoov

Kev txheeb xyuas (HPLC)

Raws li tus qauv

Ua raws

Uv max (95 feem pua ​​​​ethanol)

267,277,288nm (E1 feem pua ​​​​cm: 417, 541,416)

277nm ua

Purity (cov ntsiab lus tseem ceeb ntxiv rau isomer HPLC)

95.0 feem pua ​​~ 102.0 feem pua

98.4% ua

Xaus: nws ua raws li Enterprise tus qauv.

Tsuas yog siv rau kev lag luam lossis kev tshawb fawb, tsis yog khoom siv rau ib tus neeg twg!

 

Stability thiab cia tej yam kev mob ntawmEverolimus hmoovtseem ceeb heev. Nov yog cov ntaub ntawv ntsig txog:

Kev ruaj ntseg:

Nyob rau hauv cov xwm txheej zoo cia, nws tuaj yeem tswj kev ruaj ntseg rau lub sijhawm ntev. Nws yog qhov ruaj khov ntawm chav tsev kub tab sis tuaj yeem degrade thaum raug lub teeb, cua sov, thiab av noo. Yog li, cov hauv qab no yuav tsum tau xav txog thaum khaws cia thiab siv:

Lub teeb: nws yuav tsum tau muab khaws cia rau hauv lub teeb-resistant ntim kom tsis txhob raug tshav ntuj ncaj qha. Kev raug lub teeb ntev yuav ua rau cov tshuaj degradation.

Kub: Nws raug nquahu kom khaws cia rau hauv thaj tsam ntawm 2-8 degrees Celsius, xws li hauv lub tub yees tsis tu ncua. Tsis txhob khaws cia rau hauv qhov chaw kub thiab txias lossis nthuav tawm rau lub hnub ncaj qha.

Humidity: Nws kuj yog rhiab rau cov av noo. Nws yuav tsum tau muab khaws cia rau hauv qhov chaw qhuav thiab khaws cia rau hauv cov thawv ntim khoom kom tsis txhob ya raws qhov nkag.

Cia tej yam kev mob:

Txhawm rau kom ntseeg tau qhov zoo thiab ruaj khov, cov xwm txheej hauv qab no tuaj yeem ua raws li:

Package sealing: Khaws cia rau hauv nws qhov ntim thawj thiab xyuas kom meej tias lub hnab lossis lub raj mis tsis zoo thiab kaw zoo. Qhov no pab tiv thaiv kom tsis txhob ya raws thiab huab cua nkag.

Khaws kom deb ntawm qhov chaw tshav kub: Khaws rau hauv qhov chaw deb ntawm qhov chaw sov, tsis txhob raug tshav ntuj ncaj qha lossis ze rau cov khoom siv cua sov.

Khaws rau hauv qhov chaw qhuav: Xaiv qhov chaw qhuav thiab txias, tsis txhob muaj qhov chaw ntub dej.

Tsis txhob muaj kev vibration: Sim txo qis kev vibrations los yog cov neeg kho tshuab shocks kom tsis txhob muaj cov khoom siv lead ua tawg lossis cov khoom puas.

Cov ntaub ntawv saum toj no tsuas yog siv rau kev siv xwb, thiab qhov tshwj xeeb kev ruaj ntseg thiab kev cia khoom yuav txawv nyob ntawm cov qauv sib txawv thiab cov chaw tsim khoom.

 

Packing & shipping

Ntim:

1 ~ 2 kg

product-777-223

2-10kg

product-741-217

10-25kg

product-729-236

 

Shipping:

Tsawg dua los yog sib npaug li 50 kg

Los ntawm kev nthuav qhia qhov rooj rau qhov rooj

Fedex, DHL, UPS, TNT, EMS thiab lwm yam.

Ceev thiab yooj yim

product-179-102

50kg-200kg

Los ntawm huab cua

Ceev thiab pheej yig

product-172-94

Ntau tshaj lossis sib npaug li 200kg

Los ntawm hiav txwv

Txoj kev pheej yig tshaj

product-160-127

Los yog raws li koj yuav tsum tau xaiv txoj kev pheej yig tshaj los yog ceev.

Lub sijhawm them nyiaj

payment

Vim li cas thiaj xaiv Xi'an Yihui?

Raws li tus kws tshaj lijEverolimus APImanufacturers, peb muaj qhov zoo:

Lub zog thev naus laus zis: muaj cov cuab yeej siv tshuaj lom neeg zoo tshaj plaws thiab cov cuab yeej ntsuas kom ntseeg tau tias muaj txiaj ntsig zoo thiab muaj txiaj ntsig zoo ntawm Everolimus API.

Factory scale: muaj cov khoom siv niaj hnub thiab cov chaw tsim khoom, tuaj yeem tsim cov khoom lag luam loj thiab ua tau raws li kev xav tau ntawm kev lag luam.

Kev Tswjhwm Zoo: siv cov kev tswj xyuas nruj nruj thiab kev tshawb nrhiav kom paub tseeb tias cov khoom zoo thiab purity ua tau raws li cov qauv kev lag luam thiab cov neeg siv khoom.

Pab neeg kev paub: muaj kev nplua nuj ntau lawm thiab pab pawg kws tshaj lij, muaj peev xwm daws teeb meem hauv kev tsim khoom thiab muab kev daws teeb meem zoo.

Kev Pabcuam: tsim kom muaj kev muag khoom ua ntej, muag, thiab kev pabcuam tomqab muag los muab cov neeg siv khoom nrog txhua qhov kev pabcuam thiab kev txhawb nqa.

yihui 1

Xi 'an Yihui tuam txhab muag khoom, khoom siv ntau lawm

yihui 2

Xi'an Yihui tuam txhab muaj qib siab ntawm kev tshawb fawb thiab kev txhim kho muaj peev xwm

yihui 3

Xi 'an Yihui Company's Advanced ntau lawm cov cuab yeej thiab tshuab

yihui 4

Zoo meej kev pab cuam tom qab muag

Nyob rau hauv cov ntsiab lus, raws li ib tug kws Everolimus chaw tsim tshuaj paus, peb muaj advanced technology, scale kom zoo dua, qhov zoo tshaj plaws zoo, nplua nuj ntau lawm kev, thiab cov kev pab zoo heev. Cov txiaj ntsig zoo no yuav ua rau pebEverolimus hmoovsawv tawm hauv kev sib tw ua lag luam thiab yeej ntau tus neeg siv khoom ntseeg siab thiab kev txhawb nqa.

Cim npe nrov: Tuam Tshoj Everolimus hmoov manufacturers, lwm tus neeg, Hoobkas

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